White HS, Sarup A, Bolvig T, Kristensen AS, Petersen G, Nelson N, Pickering DS, Larsson OM, Frolund B, Krogsgaard-Larsen P, Schousboe A.
Correlation between anticonvulsant activity and inhibitory action on glial gamma-aminobutyric acid uptake of the highly selective mouse gamma-aminobutyric acid transporter 1 inhibitor 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole and its N-alkylated analogs.
J Pharmacol Exp Ther. 2002 Aug;302(2):636-44.
Brain region: cultured astrocytes
Method: Radioactive labelling